Insulin-Sensitizing Antihyperglycemic Drugs
Ali Sahin (Author)
Release Date: 2023-09-14
Insulin-sensitizing antihyperglycemic drugs are a class of medications used in the management of diabetes mellitus, particularly type 2 diabetes, by improving the body’s response to insulin. One prominent group within this category is the thiazolidinediones (TZDs), which include drugs like pioglitazone and rosiglitazone. These medications act primarily by activating peroxisome proliferator-activated receptor gamma (PPARγ) receptors, [...]
Media Type
PDF
Buy from
Price may vary by retailers
Work Type | Book Chapter |
---|---|
Published in | Current Perspective on Diabetes Mellitus in Clinical Sciences |
First Page | 115 |
Last Page | 124 |
DOI | https://doi.org/10.69860/nobel.9786053359111.10 |
ISBN | 978-605-335-911-1 (PDF) |
Language | ENG |
Page Count | 10 |
Copyright Holder | Nobel Tıp Kitabevleri |
License | https://nobelpub.com/publish-with-us/copyright-and-licensing |
Ali Sahin (Author)
Professor, Karamanoglu Mehmetbey University
https://orcid.org/0000-0003-4104-7131
Andrew J. Krentz and Clifford J. Bailey. Oral Antidiabetic Agents Current Role in Type 2 Diabetes Mellitus. Drugs 2005; 65 (3): 385-411.
Reaven GM. Role of insulin resistance in human disease. Diabetes 1988; 37: 1595-607.
Krentz AJ. Insulin resistance. Oxford: Blackwell Science, 2002.
Ginsberg HN. Insulin resistance and cardiovascular disease. J Clin Invest 2000; 106: 453-8.
Roden M. Clinical diabetes research: methods and techniques. New York: Wiley; 2007.
W. Stephen Waring. Antidiabetic drugs, Medicine 2007; 35:11.
Arrigo F.G. Cicero, Elisa Tartagni and Sibel Ertek. Metformin and its clinical use: new insights for an old drug in clinical practice. Arch Med Sci 2012; 8, 5: 907-917.
J.R. Lindsay, N.A. Duffy, A.M. McKillop, J. Ardill, F.P.M. O’Harte, P.R. Flatt and P.M. Bell. Inhibition of dipeptidyl peptidase IV activity by oral metformin in Type 2 diabetes, Diabet. Med. 22 (2005) 654-657.
Oleksandr Grytsai, Iuliia Myrgorodska, Stephane Rocchi, Cyril Ronco and Rachid Benhida. Biguanides drugs: Past success stories and promising future for drug discovery, European Journal of Medicinal Chemistry 224 (2021) 113726.
I.W. Campbell, Metformindlife begins at 50: a symposium held on the occasion of the 43rd annual meeting of the European association for the study of diabetes, amsterdam, The Netherlands, september 2007, Br. J.Diabetes
Vasc. Dis. 7 (2007) 247-252.
M. Balsells, A. García-Patterson, I. Sol_a, M. Roqu_e, I. Gich, R. Corcoy, Glibenclamide, metformin, and insulin for the treatment of gestational diabetes: a systematic review and meta-analysis, Br. Med. J. 350 (2015) h102.
C.J. Bailey, Metformin: historical overview, Diabetologia 60 (2017) 1566-1576.
Zhi-Xu He, Zhi-Wei Zhou, Yinxue Yang, Tianxin Yang, Si-Yuan Pan, Jia-Xuan Qiu and Shu-Feng Zhou. Overview of clinically approved oral antidiabetic agents for the treatment of type 2 diabetes mellitus Clinical and Experimental Pharmacology and Physiology (2015) 42, 125–138.
J.E. Gunton, P.J. Delhanty, S.-I. Takahashi, R.C. Baxter, Metformin rapidly increases insulin receptor activation in human liver and signals preferentially through insulin-receptor substrate-2, J. Clin. Endocrinol. Metabol. 88 (2003) 1323-1332.
F. Alengrin, G. Grossi, B. Canivet, J. Dolais-Kitabgi, Inhibitory effects of metformin on insulin and glucagon action in rat hepatocytes involve postreceptor alterations, Diabete Metab. 13 (1986) 591-597.
R.A. Miller, Q. Chu, J. Xie, M. Foretz, B. Viollet, M.J. Birnbaum, Biguanides suppress hepatic glucagon signalling by decreasing production of cyclic AMP, Nature 494 (2013) 256-260.
M. Stumvoll, N. Nurjhan, G. Perriello, G. Dailey, J.E. Gerich, Metabolic effects of metformin in noninsulin- dependent diabetes mellitus, N. Engl. J. Med. 333 (1995) 550-554.
Y. Fischer, J. Thomas, P. R€osen, H. Kammermeier, Action of metformin on glucose transport and glucose transporter GLUT1 and GLUT4 in heart muscle cells from healthy and diabetic rats, Endocrinology 136 (1995) 412-420.
L.S. Hermann, Metformin: a review of its pharmacological properties and therapeutic use, Diabete Metab. 5 (1979) 233-245.
Bailey CJ, Turner RC. Metformin. N Engl J Med 1996; 334:574-9.
Howlett HCS, Bailey CJ. A risk-benefi t assessment of metformin in type 2 diabetes mellitus. In: Krentz AJ, editor. Drug treatment of type 2 diabetes. Auckland: Adis Books, 2000:61-76.
Krentz AJ, Bailey CJ. Type 2 diabetes in practice. London: Royal Society of Medicine Press, 2001.
DeFronzo RA. Pharmacologic therapy for type 2 diabetes mel litus. Ann Intern Med 1999; 131: 281-30.
Scheen A. Is there a role for alpha-glucosidase inhibitors in the prevention of type 2 diabetes mellitus? Drugs 2003; 63 (10): 933-51.
Ashcroft FM, Gribble FM. ATP-sensitive K+ channels and insulin secretion: their role in health and disease. Diabetologia 1999; 42: 903-19.
Krentz AJ, Ferner RE, Bailey CJ. Comparative tolerability profi les of oral antidiabetic agents. Drug Saf 1994; 11: 223-41.
Bailey CJ, Turner RC. Metformin. N Engl J Med 1996; 334: 574-9.
Howlett HCS, Bailey CJ. A risk-benefi t assessment of metformin in type 2 diabetes mellitus. In: Krentz AJ, editor. Drug treatment of type 2 diabetes. Auckland: Adis Books, 2000: 61-76.
Sulkin T, Bosman D, Krentz AJ. Contraindications to metformin therapy in patients with NIDDM. Diabetes Care 1997; 20: 925-8.
Holt HB, Krentz AJ. Metabolic emergencies in type 2 diabetes. In: Goldstein B, M¨uller-Wieland D, editors. Textbook of type 2 diabetes. London: Martin Dunitz, 2003: 183-98.
J. Deruiter, Overview of the antidiabetic agents, Endocr. Pharmacother. Module 3 (2003) 45-50.
R.R. Koski, Oral antidiabetic agents: a comparative review, J. Pharm. Pract. 17 (2004) 39-48.
M. Rudrapal, A brief review on malaria and current antimalarial drugs, Curr. Pharma Res. 1 (2011) 286.
A.A. Soukas, H. Hao, L. Wu, Metformin as anti-aging therapy: is it for everyone? Trends Endocrinol. Metabol. 30 (2019) 745-755.
M. Antoszczak, A. Markowska, J. Markowska, A. Huczy_nski, Old wine in new bottles: drug repurposing in oncology, Eur. J. Pharmacol. 866 (2020) 172784.
A.E. Riedmaier, P. Fisel, A.T. Nies, E. Schaeffeler, M. Schwab, Metformin and cancer: from the old medicine cabinet to pharmacological pitfalls and prospects, Trends Pharmacol. Sci. 34 (2013) 126-135.
M.N. Pollak, Investigating metformin for cancer prevention and treatment: the end of the beginning, Canc. Discov. 2 (2012) 778-790.
D.R. Morales, A.D. Morris, Metformin in cancer treatment and prevention, Annu. Rev. Med. 66 (2015) 17-29.
Fürnsinn C, Waldhusl W. Thiazolidindiones: Metabolic Actions in Vitro, Diabetologia. 2002; 45: 1211-23.
Brunner LS, Suddarth DS. Textbook of Medical Surgical Nursing, 10th edition, Tahran, 2004; pp: 261-267.
Day C. Thiazolidinediones: a new class of antidiabetic drugs. Diabet Med. 1999; 16: 179-192.
Forrester MB. Pattern of thiazolidinedione exposures reported to Texas poison centers during 1998e2004. J Toxicol Environ Health 2006; 69: 2083-93.
Day C. Thiazolidinediones: a new class of antidiabetic drugs. Diabetic Med 1999; 16: 1-14
Krentz AJ, Bailey CJ, Melander A. Thiazolidinediones for type 2 diabetes. BMJ 2000; 321: 252-3
Wagstaff, A.J., Goa, K.L. (2002). Rosiglitazon: a review of its use in the management of type 2 diabetes mellitus. Drugs, 62(12):1805-1837.
Tontonoz, P., Hu, E., Spiegelman, B.M. (1994). Stimulation of adipogenesis in fi broblasts by PPARγ 2, a lipid-activated transcription factor.Cell, 79: 1147-1156.
Lopez-Lıuchı, J.V., Meıer, C.A. (1998). PPAR: from adipose tissue to the atherosclerotic plaque. European Journal of Endocrinology, 139: 363-364.
Bailey CJ, Day C. Thiazolidinediones today. Brit J Diab Vasc Dis. 2001; 1: 7-13.
Braunwald E, Fauci AS, Kasper DL, Hauser SL, Longo DL, Jameson JL. 13. Harrison İç Hastalıkları Prensipleri, Cilt 2, Nobel Kitabevleri, 2004; s: 2109-2138.
Mudaliar S, Henry RR. New oral therapies for type 2 diabetes mellitus: the glitazones or insulin sensitizers. Ann. Rev. Med. 2001; 52: 239-57.
Lebovitz HE. İnsülin resistance: defi nition and consequences. Exp. Clin. Endocrinol. Diabet. 2001; 109: 135-148.
Goldstein, B.J. Differentiating members of the thiazolidindione class: a focus on effi cacy. Diabetes Metab. Res. Rev. 2002; 18: 16-22.
Day C. Thiazolidinediones: a new class of antidiabetic drugs. Diabet Med. 1999; 16: 179-192.
Fürnsinn C, Waldhusl W. Thiazolidindiones: Metabolic Actions in Vitro, Diabetologia. 2002; 45: 1211-23.
Brunner LS, Suddarth DS. Textbook of Medical Surgical Nursing, 10th edition, Tahran, 2004; pp: 261-267.
Baldwin SJ, Clarke SE, Chenery RJ. Characterisation of the cytochrome P450 enzymes involved in the in vitro metabolism of rosiglitazone. Br J Clin Pharmacol 1999; 48: 424-32.
Forrester MB. Pattern of thiazolidinedione exposures reported toTexas poison centers during 1998e2004. J Toxicol Environ Health 2006; 69: 2083-93.
W Stephen Waring. Antidiabetic drugs, Medicine 2016, 44;3:138-140.
Yki-Ja¨rvinen H. Thiazolidinedions. N Engl J Med 2004; 351:1106-18.
Parulkar AA, Pendergrass ML, Granda-Ayala R, et al. Nonhypoglycemic effects of thiazolidinediones. Ann Intern Med 2001; 134: 61-71.
Marten FMAC, Visseren FLJ, Lemay J, et al. Metabolic and additional vascular effects of thiazolidinediones. Drugs 2002;62 (10): 1463-80.
Buchanan TA, Xiang AH, Peters RK, et al. Preservation of pancreatic beta-cell function and prevention of type 2 diabetes by pharmacological treatment of insulin resistance in high-risk hispanic women. Diabetes 2002; 51: 2796-803.
Viral S. Jain, Dhagash K. Vora, C. S. Ramaa. Thiazolidine-2,4-diones: Progress towards multifarious applications. Bioorganic & Medicinal Chemistry 21 (2013) 1599–1620
onix_3.0::thoth | Thoth ONIX 3.0 |
---|---|
onix_3.0::project_muse | Project MUSE ONIX 3.0 |
onix_3.0::oapen | OAPEN ONIX 3.0 |
onix_3.0::jstor | JSTOR ONIX 3.0 |
onix_3.0::google_books | Google Books ONIX 3.0 |
onix_3.0::overdrive | OverDrive ONIX 3.0 |
onix_2.1::ebsco_host | EBSCO Host ONIX 2.1 |
csv::thoth | Thoth CSV |
json::thoth | Thoth JSON |
kbart::oclc | OCLC KBART |
bibtex::thoth | Thoth BibTeX |
doideposit::crossref | CrossRef DOI deposit |
onix_2.1::proquest_ebrary | ProQuest Ebrary ONIX 2.1 |
marc21record::thoth | Thoth MARC 21 Record |
marc21markup::thoth | Thoth MARC 21 Markup |
marc21xml::thoth | Thoth MARC 21 XML |